Preparation of 10-keto morphinans by benzylic oxidation
The present invention provides processes for the preparation of 10-keto and/or 10-hydroxy morphinans. In particular, the invention provides to processes for preparing a 10-keto morphinan by chromium-catalyzed benzylic oxidation of a morphinan with a periodic acid.
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Main Authors | , , , |
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Format | Patent |
Language | English |
Published |
20.11.2012
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Online Access | Get full text |
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Summary: | The present invention provides processes for the preparation of 10-keto and/or 10-hydroxy morphinans. In particular, the invention provides to processes for preparing a 10-keto morphinan by chromium-catalyzed benzylic oxidation of a morphinan with a periodic acid. |
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