DIBENZOFURANCARBOXAMIDES

This invention is directed to certain dibenzofurancarboxamides and their use as 5HT3? antagonists having unique CNS, anti-emetic and gastric prokinetic activity void of any significant D2? receptor binding properties. This invention also describes novel processes necessary for their perparation. L&#...

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Bibliographic Details
Main Authors KUHLA, DONALD, E, AIREY, JOHN, EDWARD, CAMPBELL, HENRY, F, KLEIN, SCOTT, IRA, POWERS, MATTHEW, RAY, YOUSSEFYEH, RAYMOND, D
Format Patent
LanguageEnglish
Published 02.11.1989
Edition4
Subjects
CHEMISTRY
HETEROCYCLIC COMPOUNDS
HUMAN NECESSITIES
HYGIENE
MEDICAL OR VETERINARY SCIENCE
METALLURGY
ORGANIC CHEMISTRY
PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS
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Summary:This invention is directed to certain dibenzofurancarboxamides and their use as 5HT3? antagonists having unique CNS, anti-emetic and gastric prokinetic activity void of any significant D2? receptor binding properties. This invention also describes novel processes necessary for their perparation. L'invention concerne certains dibenzofurancarboxamides et leur utilisation comme antagonistes des 5HT3, ayant une activité CNS, anti-émétique et procinétique gastrique unique dépourvue de toutes propriétés significatives de liaison du récepteur D2. Cette invention concerne également de nouveaux procédés nécessaires à leur préparation.
Bibliography:Application Number: WO1989US01739