QUINAZOLINE COMPOUND AND APPLICATION THEREOF

A quinazoline compound and an application thereof. The quinazoline compound is shown as a formula 1, it has a good inhibiting effect on KRAS G12D mutant protein and has a good patent medicine prospect. L'invention concerne un composé de quinazoline et une application de celui-ci. Le composé de...

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Bibliographic Details
Main Authors ZHANG, Chaoxin, HUO, Guoyong, WANG, Xuesong, MAO, Haibin, FU, Yuhong, XIA, Guangxin, LI, Zhilong, KE, Ying, MA, Xing
Format Patent
LanguageChinese
English
French
Published 06.07.2023
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Summary:A quinazoline compound and an application thereof. The quinazoline compound is shown as a formula 1, it has a good inhibiting effect on KRAS G12D mutant protein and has a good patent medicine prospect. L'invention concerne un composé de quinazoline et une application de celui-ci. Le composé de quinazoline est représenté par la formule 1, il a un bon effet d'inhibition sur la protéine mutante KRAS G12D et a une bonne perspective de médicament breveté. 一种喹唑啉类化合物及其应用。喹唑啉类化合物如式1所示,其对KRAS G12D突变蛋白具有良好的抑制作用,有良好的成药前景。
Bibliography:Application Number: WO2022CN144234