SYNTHESIS OF 1,2,5-TRI-0-BENZ0YL-3-DIBENZYLAMIN0-3-DE0XYRIB0SE AS INTERMEDIATE FOR PRODUCING 3'-AMINO-3'-DEOXYADENOSINE AND 3'-AMINO-3'-DEOXYGUANOSINE AND THE PROTECTED DERIVATIVES THEREOF

The invention generally relates to improved processes for the preparation of intermediates of a cyclic dinucleotide which is useful as a STING agonist. L'invention concerne de manière générale des procédés améliorés pour la préparation d'intermédiaires d'un dinucléotide cyclique qui e...

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Main Authors YUAN, Changxia, WU, Shulin, ZHONGMIN, Xu, YU, Miao, SCHMIDT, Michael Anthony, ROGERS, Amanda J, ZHU, Jason J, SIMMONS, Eric M, ORTIZ, Adrian
Format Patent
LanguageEnglish
French
Published 13.08.2020
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Summary:The invention generally relates to improved processes for the preparation of intermediates of a cyclic dinucleotide which is useful as a STING agonist. L'invention concerne de manière générale des procédés améliorés pour la préparation d'intermédiaires d'un dinucléotide cyclique qui est utile en tant qu'agoniste de STING.
Bibliography:Application Number: WO2020US16694