α-AMINO ACRYLATE MICROBICIDE, AND PREPARATION METHOD THEREFOR AND USES THEREOF

• Main Authors: XUE, Jing, YANG, Huaipu, FAN, Zhijin, JIN, Jianyu, MA, Liuyong, YU, Bin, WU, Qifan, HAN, Cenhui, WU, Aoben, ZHANG, Nailou, QIAN, Xiaolin, WANG, Haixia
• Format: Patent
• Language: Chinese; English; French
• Published: 22.11.2018
• Subjects: AGRICULTURE; ANIMAL HUSBANDRY; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES, AS HERBICIDES; CHEMISTRY; FISHING; FORESTRY; HETEROCYCLIC COMPOUNDS; HUMAN NECESSITIES; HUNTING; METALLURGY; ORGANIC CHEMISTRY; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS; PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTSTHEREOF; TRAPPING

Provided are an α-amino acrylate microbicide, and a preparation method therefor and uses thereof. Based on the principle of pesticide molecular design, the structural reform of the agricultural anti-plant virus activity is carried on lead compounds having the medical anti-coronavirus activity, and a series of α-amino-acrylic derivatives are designed and synthesized, and in particular, α-amino acrylic derivatives containing piperidine rings are synthesized, and the systematic biological activity screening is carried by using known compounds as positive control compounds, which provides many effective anti-virus leading molecules for the preparation of pesticides, and has positive significance to the reduced use of f pesticides and the protection of environmental ecology. L'invention concerne un microbicide α-amino acrylate, son procédé de préparation et ses utilisations. Sur la base du principe de la conception moléculaire de pesticides, la réforme structurale de l'activité antivirale des végétaux est effectué