AZAINDOLE DERIVATIVES AND THEIR USE AS ERK KINASE INHIBITORS

The present invention concerns a compound of formula (I): H or one of its pharmaceutically acceptable salts, especially for use as inhibitors of the ERK kinase activity in particular ERK2 activity, it also concerns prodrugs of these compounds. La présente invention concerne un composé de formule (I)...

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Bibliographic Details
Main Authors GUICHOU, Jean-François, GEOFFROY, Clément, GELIN, Muriel, BORIES, Cédric, DUQUENNE, Charline, LABESSE, Gilles, BESSIN, Yannick
Format Patent
LanguageEnglish
French
Published 26.05.2017
Subjects
CHEMISTRY
HETEROCYCLIC COMPOUNDS
HUMAN NECESSITIES
HYGIENE
MEDICAL OR VETERINARY SCIENCE
METALLURGY
ORGANIC CHEMISTRY
PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS
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Summary:The present invention concerns a compound of formula (I): H or one of its pharmaceutically acceptable salts, especially for use as inhibitors of the ERK kinase activity in particular ERK2 activity, it also concerns prodrugs of these compounds. La présente invention concerne un composé de formule (I) ou un de ses sels pharmaceutiquement acceptables, notamment en tant qu'inhibiteurs de l'activité kinase ERK en particulier l'activité ERK2. L'invention concerne également des promédicaments de ces composés.
Bibliography:Application Number: WO2016EP78080