SOLID STATE FORMS OF ELUXADOLINE

Disclosed are solid state forms of Eluxadoline, processes for their preparations, compositions comprising them and their medical use. The present invention also encompasses solid state forms of Eluxadoline for use in the preparation of other solid state forms of Eluxadoline, particularly form alpha....

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Main Authors MUSANIC, Sanja, Matecic, LEKSIC, Edislav, MARINKOVIC, Marina, VUSAK, Vitomir
Format Patent
LanguageEnglish
French
Published 26.01.2017
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Summary:Disclosed are solid state forms of Eluxadoline, processes for their preparations, compositions comprising them and their medical use. The present invention also encompasses solid state forms of Eluxadoline for use in the preparation of other solid state forms of Eluxadoline, particularly form alpha. L'invention concerne des formes à l'état solide d'Éluxadoline, des procédés pour leurs préparations, des compositions les comprenant et leur utilisation médicale. La présente invention concerne également des formes à l'état solide d'Éluxadoline à utiliser dans la préparation d'autres formes à l'état solide d'Éluxadoline, en particulier de forme alpha.
Bibliography:Application Number: WO2016US43678