CATHEPSIN CYSTEINE PROTEASE INHIBITORS

This invention relates to a novel class of compounds which are cysteine protease inhibitors, including but not limited to, inhibitors of cathepsins K, L, S and B. These compounds are useful for treating diseases in which inhibition of bone resorption is indicated, such as osteoporosis. La présente i...

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Main Authors XU, SHIMIN, PAONE, DANIEL, V, FU, JIANMIN, STACHEL, SHAWN, GINNETTI, ANTHONY, LI, JING, LIM, JOHN
Format Patent
LanguageEnglish
French
Published 16.04.2015
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Summary:This invention relates to a novel class of compounds which are cysteine protease inhibitors, including but not limited to, inhibitors of cathepsins K, L, S and B. These compounds are useful for treating diseases in which inhibition of bone resorption is indicated, such as osteoporosis. La présente invention concerne une nouvelle classe de composés qui sont des inhibiteurs de protéases à cystéine, comprenant entre autres, des inhibiteurs de cathepsines K, L, S et B. Ces composés sont utiles pour le traitement de maladies, telles que l'ostéoporose, dans lesquelles l'inhibition de la résorption osseuse est indiquée.
Bibliography:Application Number: WO2014US58934