MANUFACTURING PROCESS FOR PYRIMIDINE DERIVATIVES
The invention relates to processes for manufacturing a compound of formula (5) or a stereoisomer, tautomer or a salt thereof, wherein the substituents are as defined in the specification. The invention further relates to new manufacturing processes for specific solid forms of Compound A and its salt...
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| Main Authors | , , , , , , , , , , |
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| Format | Patent |
| Language | English French |
| Published |
05.04.2012
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| Subjects | |
| Online Access | Get full text |
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| Abstract | The invention relates to processes for manufacturing a compound of formula (5) or a stereoisomer, tautomer or a salt thereof, wherein the substituents are as defined in the specification. The invention further relates to new manufacturing processes for specific solid forms of Compound A and its salts, to such solid forms and to use of said solid forms for the therapeutic treatment of warm-blooded animals.
La présente invention a pour objet des procédés de fabrication d'un composé de formule 5 ou de l'un de stéréoisomères, tautomères ou sels, dans laquelle les substituants sont tels que définis dans le mémoire. L'invention a en outre pour objet de nouveaux procédés de fabrication de formes solides spécifiques du composé A et de ses sels, lesdites formes solides et l'utilisation desdites formes solides pour le traitement thérapeutique d'animaux à sang chaud. |
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| AbstractList | The invention relates to processes for manufacturing a compound of formula (5) or a stereoisomer, tautomer or a salt thereof, wherein the substituents are as defined in the specification. The invention further relates to new manufacturing processes for specific solid forms of Compound A and its salts, to such solid forms and to use of said solid forms for the therapeutic treatment of warm-blooded animals.
La présente invention a pour objet des procédés de fabrication d'un composé de formule 5 ou de l'un de stéréoisomères, tautomères ou sels, dans laquelle les substituants sont tels que définis dans le mémoire. L'invention a en outre pour objet de nouveaux procédés de fabrication de formes solides spécifiques du composé A et de ses sels, lesdites formes solides et l'utilisation desdites formes solides pour le traitement thérapeutique d'animaux à sang chaud. |
| Author | MICHEL, PASCAL WAYKOLE, LILADHAR MURLIDHAR TESTA, MARIA CATERINA FLUBACHER, DIETMAR CALIENNI, JOHN VINCENT LIU, HUI MOSE, RASMUS DE LA CRUZ, MARILYN KARPINSKI, PIOTR H KAPA, PRASAD KOTESWARA GONG, BAOQING |
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| DocumentTitleAlternate | PROCÉDÉ DE FABRICATION DE DÉRIVÉS DE PYRIMIDINE |
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| RelatedCompanies | MICHEL, PASCAL WAYKOLE, LILADHAR MURLIDHAR TESTA, MARIA CATERINA FLUBACHER, DIETMAR CALIENNI, JOHN VINCENT LIU, HUI MOSE, RASMUS DE LA CRUZ, MARILYN KARPINSKI, PIOTR H NOVARTIS AG KAPA, PRASAD KOTESWARA GONG, BAOQING |
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| Title | MANUFACTURING PROCESS FOR PYRIMIDINE DERIVATIVES |
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