NOVEL HETEROARYL DERIVATIVE

A highly effective FAAH inhibitor, and especially a prophylactic or drug for severe pain, which can be administered orally, are needed. Provided is a pharmaceutical composition having as an active ingredient a novel heteroaryl derivative or salt as represented by formula (I) below and a solvate ther...

Full description

Saved in:
Bibliographic Details
Main Authors KAMINO TOMOYUKI, MIZUNO TAKASHI, NAGASUE HIROSHI
Format Patent
LanguageEnglish
French
Japanese
Published 01.09.2011
Subjects
CHEMISTRY
HETEROCYCLIC COMPOUNDS
HUMAN NECESSITIES
HYGIENE
MEDICAL OR VETERINARY SCIENCE
METALLURGY
ORGANIC CHEMISTRY
PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS
Online AccessGet full text

Cover

More Information
Summary:A highly effective FAAH inhibitor, and especially a prophylactic or drug for severe pain, which can be administered orally, are needed. Provided is a pharmaceutical composition having as an active ingredient a novel heteroaryl derivative or salt as represented by formula (I) below and a solvate thereof. Said pharmaceutical composition can be used especially as an FAAH inhibitor or as a prophylactic or drug for severe pain. L'invention porte sur un inhibiteur de FAAH extrêmement efficace et notamment sur un agent prophylactique ou sur un médicament pour la douleur sévère, qui peut être administré par voie orale. L'invention décrit une composition pharmaceutique qui possède, comme principe actif, un nouveau dérivé hétéroaryle ou un sel, tel que représenté dans la formule (I) ci-dessous, et un solvate de celui-ci. Ladite composition pharmaceutique peut être utilisée notamment comme inhibiteur de FAAH ou en tant qu'agent prophylactique ou médicament pour la douleur sévère.
Bibliography:Application Number: WO2011JP54366