SYNTHESIS OF SUBSTITUTED PYRAZOLINE CARBOXAMIDINE DERIVATIVES

This invention relates to organic chemistry, in particular to processes for the preparation of pyrazoline carboxamidine derivatives of formula (I), known as potent 5-HT6 antagonists. The invention also relates to novel intermediates of these compounds. wherein the symbols have the meanings given in...

Full description

Saved in:
Bibliographic Details
Main Authors LANGE, JOSEPHUS H.M, DEN HARTOG, ARNOLD P, VAN LOEVEZIJN, ARNOLD, BARF, GERRIT A
Format Patent
LanguageEnglish
French
Published 07.09.2012
Subjects
CHEMISTRY
HETEROCYCLIC COMPOUNDS
METALLURGY
ORGANIC CHEMISTRY
Online AccessGet full text

Cover

More Information
Summary:This invention relates to organic chemistry, in particular to processes for the preparation of pyrazoline carboxamidine derivatives of formula (I), known as potent 5-HT6 antagonists. The invention also relates to novel intermediates of these compounds. wherein the symbols have the meanings given in the description. La présente invention concerne la chimie organique, en particulier des procédés de préparation de dérivés de pyrazoline carboxamidine de formule (I), connus pour être de puissants antagonistes de 5-HT6. L'invention concerne également de nouveaux intermédiaires de ces composés. Les symboles ont la signification donnée dans la description.
Bibliography:Application Number: WO2011EP51100