N-(HETERO)ARYL-PYRROLIDINE DERIVATIVES OF PYRAZOL-4-YL-PYRROLO[2,3-d]PYRIMIDINES AND PYRROL-3-YL-PYRROLO[2,3-d]PYRIMIDINES AS JANUS KINASE INHIBITORS
The present invention relates to N-(hetero)aryl-pyrrolidine derivatives of Formula (I): which are JAK inhibitors, such as selective JAK1 inhibitors, useful in the treatment of JAK-associated diseases including, for example, inflammatory and autoimmune disorders, as well as cancer. La présente invent...
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Main Authors | , , , , , , , , |
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Format | Patent |
Language | English French |
Published |
25.11.2010
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Subjects | |
Online Access | Get full text |
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Summary: | The present invention relates to N-(hetero)aryl-pyrrolidine derivatives of Formula (I): which are JAK inhibitors, such as selective JAK1 inhibitors, useful in the treatment of JAK-associated diseases including, for example, inflammatory and autoimmune disorders, as well as cancer.
La présente invention concerne des dérivés N-(hétéro)aryl-pyrrolidine de formule (I) : qui sont des inhibiteurs JAK, tels que des inhibiteurs JAK1 sélectifs. Ces inhibiteurs sont utiles dans le traitement de maladies associées à la JAK, comprenant par exemple les affections inflammatoires et les maladies auto-immunes, ainsi que le cancer. |
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Bibliography: | Application Number: WO2010US35783 |