4-AMINOTHIENO[2,3-d]PYRIMIDINE-6-CARBONITRILE DERIVATIVES AS PDE7 INHIBITORS
New 4-aminothieno[2,3-d]pyrimidine-6-carbonitrile derivatives having the chemical structure of general formula (I), and pharmaceutically acceptable salts thereof are disclosed as well as processes for their preparation and to pharmaceutical compositions containing them and their use in the treatment...
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| Main Authors | , , , , |
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| Format | Patent |
| Language | English French |
| Published |
05.08.2004
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| Edition | 7 |
| Subjects | |
| Online Access | Get full text |
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| Abstract | New 4-aminothieno[2,3-d]pyrimidine-6-carbonitrile derivatives having the chemical structure of general formula (I), and pharmaceutically acceptable salts thereof are disclosed as well as processes for their preparation and to pharmaceutical compositions containing them and their use in the treatment, prevention or suppression of pathological conditions, diseases and disorders susceptible of being improved by inhibition of PDE7.
L'invention concerne des dérivés de 4-aminothiéno[2,3-d]pyrimidine-6-carbonitrile présentant la structure chimique de formule générale (I), des sels acceptables sur le plan pharmaceutique de ceux-ci, des procédés de préparation de ceux-ci et des compositions pharmaceutiques renfermant ceux-ci, ainsi que l'utilisation de celles-ci dans le traitement, la prévention ou la suppression d'états pathologiques, de maladies et de troubles susceptibles d'être améliorés par l'inhibition de PDE7. |
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| AbstractList | New 4-aminothieno[2,3-d]pyrimidine-6-carbonitrile derivatives having the chemical structure of general formula (I), and pharmaceutically acceptable salts thereof are disclosed as well as processes for their preparation and to pharmaceutical compositions containing them and their use in the treatment, prevention or suppression of pathological conditions, diseases and disorders susceptible of being improved by inhibition of PDE7.
L'invention concerne des dérivés de 4-aminothiéno[2,3-d]pyrimidine-6-carbonitrile présentant la structure chimique de formule générale (I), des sels acceptables sur le plan pharmaceutique de ceux-ci, des procédés de préparation de ceux-ci et des compositions pharmaceutiques renfermant ceux-ci, ainsi que l'utilisation de celles-ci dans le traitement, la prévention ou la suppression d'états pathologiques, de maladies et de troubles susceptibles d'être améliorés par l'inhibition de PDE7. |
| Author | MINGUEZ ORTEGA, JOSE, MIGUEL ALVAREZ-BUILLA GOMEZ, JULIO TERRICABRAS BELART, EMMA SEGARRA MATAMOROS, VICTOR, MANUEL VAQUERO LOPEZ, JUAN, JOSE |
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| DocumentTitleAlternate | DERIVES DE 4-AMINOTHIENO[2,3-D]PYRIMIDINE-6-CARBONITRILE UTILISES COMME INHIBITEURS DE PDE7 |
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| RelatedCompanies | MINGUEZ ORTEGA, JOSE, MIGUEL ALVAREZ-BUILLA GOMEZ, JULIO ALMIRALL PRODESFARMA S.A TERRICABRAS BELART, EMMA SEGARRA MATAMOROS, VICTOR, MANUEL VAQUERO LOPEZ, JUAN, JOSE |
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| Title | 4-AMINOTHIENO[2,3-d]PYRIMIDINE-6-CARBONITRILE DERIVATIVES AS PDE7 INHIBITORS |
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