ANTIBACTERIAL HAVING PYRAZOLE SKELETON

A compound which has a pyrazole skeleton and has excellent antibacterial activity against gram-positive bacteria and resistant gram-positive bacteria. The compound having a pyrazole skeleton is represented by the following formula (I): (I) wherein R1 is lower alkyl; R2 is hydrogen or lower alkyl; R3...

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Main Authors HARA, HIROTO, YOSHIDA, TOSHIO, YOKOSE, KAZUTERU, YASUDA, MINORU, NAKASHIMA, MIHOKO, IKESUE, KOICHI, MAEDA, YUTAKA
Format Patent
LanguageEnglish
French
Japanese
Published 15.04.2004
Edition7
Subjects
CHEMISTRY
HETEROCYCLIC COMPOUNDS
HUMAN NECESSITIES
HYGIENE
MEDICAL OR VETERINARY SCIENCE
METALLURGY
ORGANIC CHEMISTRY
PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS
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Summary:A compound which has a pyrazole skeleton and has excellent antibacterial activity against gram-positive bacteria and resistant gram-positive bacteria. The compound having a pyrazole skeleton is represented by the following formula (I): (I) wherein R1 is lower alkyl; R2 is hydrogen or lower alkyl; R3 is phenyl or benzyl; and X is hydrogen or a group represented by the following formula, (II) L'invention porte sur un composé à squelette de pyrazole et à excellente activité bactéricide contre les bactéries gram-positives et en particulier les bactéries gram-positives résistantes. Ledit composé présente la formule (I) dans laquelle: R1 est alkyle inférieur, R2 est H ou alkyle inférieur, R3 est phényle ou benzyle, et X est H ou un groupe de formule (II).
Bibliography:Application Number: WO2002JP10367