Process for the preparation cabazitaxel

The present invention discloses a process for the preparation of 4-acetoxy-2α-benzoyloxy-5 ,20-epoxy-1-hydroxy-7 ,10 -dimethoxy-9-oxotax-11-en-13α-yl(2R,3S)-3-tert-butoxycarbonylamino-2-hydroxy-3-phenyl-propionate Cabazitaxel (I).

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Bibliographic Details
Main Authors LAHIRI SASWATA, AZIM ABUL, PANDA NILENDU, GUPTA NITIN, MISHRA BHUWAN BHASKAR, SANGHANI SUNIL
Format Patent
LanguageEnglish
Published 02.12.2014
Subjects
ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAININGELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN,SULFUR, SELENIUM OR TELLURIUM
CHEMISTRY
HETEROCYCLIC COMPOUNDS
METALLURGY
ORGANIC CHEMISTRY
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Summary:The present invention discloses a process for the preparation of 4-acetoxy-2α-benzoyloxy-5 ,20-epoxy-1-hydroxy-7 ,10 -dimethoxy-9-oxotax-11-en-13α-yl(2R,3S)-3-tert-butoxycarbonylamino-2-hydroxy-3-phenyl-propionate Cabazitaxel (I).
Bibliography:Application Number: US201213625155