Intermediaties for aminooxypyrrolidinylthiocarbapenem compounds

An antibacterial aminooxypyrrolidinylthiocarbapenem I, its production from the corresponding carbapenem V and thiol VI, its pharmaceutical formulation, and its use for combating bacteria are presented. I V VI (wherein R is optionally substituted amino; R1 is hydrogen or 1C to 5C alkyl; R2 is hydroge...

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Bibliographic Details
Main Authors SENDO; YUJI, KII; MAKOTO
Format Patent
LanguageEnglish
Published 04.06.1996
Edition6
Subjects
CHEMISTRY
HETEROCYCLIC COMPOUNDS
HUMAN NECESSITIES
HYGIENE
MEDICAL OR VETERINARY SCIENCE
METALLURGY
ORGANIC CHEMISTRY
PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS
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Summary:An antibacterial aminooxypyrrolidinylthiocarbapenem I, its production from the corresponding carbapenem V and thiol VI, its pharmaceutical formulation, and its use for combating bacteria are presented. I V VI (wherein R is optionally substituted amino; R1 is hydrogen or 1C to 5C alkyl; R2 is hydrogen or a conventional hydroxy protective group; R3 is hydrogen or an imino protective group or imino substituent; R4 is 1C to 5C alkylene; and R5 is hydrogen or a conventional carboxy protective group; X is a leaving group; R6 is hydrogen or a thiol protective group; and wavy lines each shows a bond in R or S configuration).
Bibliography:Application Number: US19940273979