TETRAHYDROQUINOLINE COMPOUNDS CONTAINING CYANOMETHYLIDINE AND BENZOICSULFIMIDO GROUPS
A procedure for the preparation of antibacterial agents of the formula **(See formula)** where R represents **(See formula)** R1, R2 and R3 each represent hydrogen, nitro, lower alkyl, dialkyl lower amino, alkanoyl (lower) amino, amino, hydroxyl, alkanoyl (lower) -oxy, lower alkyl, lower alkoxy, sul...
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Main Authors | , |
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Format | Patent |
Language | English |
Published |
27.07.1971
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Subjects | |
Online Access | Get full text |
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Summary: | A procedure for the preparation of antibacterial agents of the formula **(See formula)** where R represents **(See formula)** R1, R2 and R3 each represent hydrogen, nitro, lower alkyl, dialkyl lower amino, alkanoyl (lower) amino, amino, hydroxyl, alkanoyl (lower) -oxy, lower alkyl, lower alkoxy, sulfamyl., chlorine, iodine, bromine, fluorine, or trifluoromethyl and the non-toxic and pharmaceutically acceptable salts thereof; whose procedure is to react a compound of formula **(See formula)** where R is the one defined above, or one of its non-toxic and pharmaceutically acceptable salts, with a guanylcarbamoylation agent, in the presence of a base, at a pH higher than 6 and at a temperature between approximately -20ºC and 50ºC. (Machine-translation by Google Translate, not legally binding) |
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Bibliography: | Application Number: USD3595863 |