PROCESSES FOR THE PREPARATION OF (S)-2-(4-CHLORO-2-METHOXYPHENYL)-2-((3 -METHOXY-5-(M ETHYLSULFONYL)PHENYL)AMINO)-1 -(1H-INDOL-3-YL)ETHENONE DERIVATIVES

The present invention relates to novel chiral synthesis of mono- or di-substituted indole compounds of formula (I)wherein:R1 is H, R2 is F and R3 is H or CH3,R1 is H, CH3 or F, R2 is OCH3 and R3 is H andR1 is H, R2 is OCH3 and R3 is CH3,R1 is CH3, R2 is F and R3 is H,R1 is CF3 or OCF3, R2 is H and R...

Full description

Saved in:
Bibliographic Details
Main Authors Wu, Kai, Eriksson, Carl Arne Magnus, Oost, Rik, Schweitzer-Chaput, Bertrand, Coesemans, Erwin
Format Patent
LanguageEnglish
Published 19.09.2024
Subjects
ACYCLIC OR CARBOCYCLIC COMPOUNDS
CHEMISTRY
HETEROCYCLIC COMPOUNDS
METALLURGY
ORGANIC CHEMISTRY
Online AccessGet full text

Cover

More Information
Summary:The present invention relates to novel chiral synthesis of mono- or di-substituted indole compounds of formula (I)wherein:R1 is H, R2 is F and R3 is H or CH3,R1 is H, CH3 or F, R2 is OCH3 and R3 is H andR1 is H, R2 is OCH3 and R3 is CH3,R1 is CH3, R2 is F and R3 is H,R1 is CF3 or OCF3, R2 is H and R3 is H,R1 is OCF3, R2 is OCH3 and R3 is H andR1 is OCF3, R2 is H and R3 is CH3.
Bibliography:Application Number: US202218571817