SARS-COV-2 MPRO INHIBITOR COMPOUNDS

The invention described herein relates to compounds of Formula (1b):or a salt thereof, wherein R1, R1a, R2, R3 and R5 are defined herein, and their use in the treatment of SARS-CoV-2 and related viruses and disorders associated with SARS-CoV-2.

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Main Authors PICKWORTH, Mark, DE GRAAF, Chris, HIGUERUELO, Alicia Perez, CONGREVE, Miles Stuart, CHRISTOPHER, John Andrew, MASON, Jonathan Stephen
Format Patent
LanguageEnglish
Published 04.07.2024
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Abstract The invention described herein relates to compounds of Formula (1b):or a salt thereof, wherein R1, R1a, R2, R3 and R5 are defined herein, and their use in the treatment of SARS-CoV-2 and related viruses and disorders associated with SARS-CoV-2.
AbstractList The invention described herein relates to compounds of Formula (1b):or a salt thereof, wherein R1, R1a, R2, R3 and R5 are defined herein, and their use in the treatment of SARS-CoV-2 and related viruses and disorders associated with SARS-CoV-2.
Author CONGREVE, Miles Stuart
MASON, Jonathan Stephen
PICKWORTH, Mark
DE GRAAF, Chris
HIGUERUELO, Alicia Perez
CHRISTOPHER, John Andrew
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– fullname: MASON, Jonathan Stephen
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Snippet The invention described herein relates to compounds of Formula (1b):or a salt thereof, wherein R1, R1a, R2, R3 and R5 are defined herein, and their use in the...
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SubjectTerms CHEMISTRY
HETEROCYCLIC COMPOUNDS
HUMAN NECESSITIES
HYGIENE
MEDICAL OR VETERINARY SCIENCE
METALLURGY
ORGANIC CHEMISTRY
PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
Title SARS-COV-2 MPRO INHIBITOR COMPOUNDS
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