PTERIDINES AND THEIR USE AS AGROCHEMICALS

• Main Authors: BREWSTER WILLIAM K, LOWE CHRISTIAN T, RIEDER BRENT J, KLITTICH CARLA J.R, DEMETER DAVID A, YERKES CARLA N, YAO CHENGLIN, ERICKSON W. RANDAL, NUGENT JAIME S, SIDDALL THOMAS L, ZHU YUANMING
• Format: Patent
• Language: English
• Published: 26.09.2013
• Subjects: AGRICULTURE; ANIMAL HUSBANDRY; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES, AS HERBICIDES; FISHING; FORESTRY; HUMAN NECESSITIES; HUNTING; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS; PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTSTHEREOF; TRAPPING

The present disclosure relates to 1- or 2-(4-(aryloxy)-phenyl)ethylamino-, oxy- or sulfanyl)pteridines and 1- or 2-(4-(heteroaryloxy)-phenyl)ethylamino-, oxy- or sulfanyl)pteridines and their use as agrochemicals and animal health products. More specifically, the invention provides new compounds of the formula (I-A): wherein: R is H CH3, phenyl, or a heterocycle comprising a 5 or 6 membered single ring or a fused ring system comprising at least one 5 or 6 membered heterocycle optionally substituted with H, halo, lower alkyl, lower alkoxy, benzyloxy, lower alkenyl, lower alkynyl, haloalkyl, haloalkoxy, NO2, CN, lower alkoxycarbonyl, lower alkylcarbonyl, lower alkyl-SOq, and aldoximes and lower alkyloximes, optionally substituted on oxygen by lower alkyl. Z is H, a C-C single bond, CH2, NH, O, S, CN, CH2O, OCH2, CH2CH2O, or OCH2CH2; m is 4; p is 0 or 1; q is an integer from 0 to 2; R1 is independently H, halo, lower alkyl, lower alkenyl, lower alkynyl, hydroxy, lower alkoxy, haloalkyl, haloalkoxy, NO2, CN, lower alklycarbonyl, lower alkoxycarbonyl, mercapto, lower alkylthio, aldoximes and lower alkyloximes, optionally substituted on oxygen by lower alkyl; Y is a C-C single bond, C(R5n)O or C(R5n); n is 2.