Process for the preparation of Crisaborole in a stable crystal form

The present invention relates to a process for the preparation of crisaborole of formula (I):by preparing intermediates of formulas (II) and (III):

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Bibliographic Details
Main Authors Gassa, Federico, Quaroni, Marco, Sada, Mara, Bertolini, Giorgio, Feliciani, Lazzaro, Mazza, Alberto
Format Patent
LanguageEnglish
Published 10.05.2022
Subjects
ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAININGELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN,SULFUR, SELENIUM OR TELLURIUM
CHEMISTRY
METALLURGY
ORGANIC CHEMISTRY
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Summary:The present invention relates to a process for the preparation of crisaborole of formula (I):by preparing intermediates of formulas (II) and (III):
Bibliography:Application Number: US202016926370