13-substituted milbemycin derivatives, their preparation and their use against insects and other pests

Compounds of formula (I) and salts thereof: wherein: R1 represents methyl, ethyl, isopropyl or s-butyl; R2 represents hydrogen or alkyl; R3 represents hydrogen, optionally substituted alkanoyl, optionally substituted alkenoyl, optionally substituted alkynoyl, alkylsulfonyl, or alkoxycarbonyl, or R2...

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Bibliographic Details
Main Authors SAITO, AKIO, SUGIYAMA, YOKO, TOYAMA, TOSHIMITSU, NANBA, TOSHIHIKO
Format Patent
LanguageEnglish
Published 11.08.2007
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Summary:Compounds of formula (I) and salts thereof: wherein: R1 represents methyl, ethyl, isopropyl or s-butyl; R2 represents hydrogen or alkyl; R3 represents hydrogen, optionally substituted alkanoyl, optionally substituted alkenoyl, optionally substituted alkynoyl, alkylsulfonyl, or alkoxycarbonyl, or R2 and R3 together with the nitrogen atom to which they are attached form a saturated, optionally substituted 4- to 6-membered heterocyclic ring group; and the moiety -a- together with the carbon atom to which it is attached forms a 3- to 6-membered cycloalkyl group. These compounds have anthelmintic, acaricidal and insecticidal activity.
Bibliography:Application Number: TW200190109990