Novel benzoxazine benzimidazol derivatives, pharmaceutical composition comprising same, and use thereof

The present invention relates to a novel benzoxazine benzimidazole derivative of formula (1) as an antagonist against a vanilloid receptor-1, a pharmaceutical composition comprising the same as an active ingredient, and a use thereof. The benzoxazine benzimidazole derivative of the present invention...

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Main Authors HYUN, HYAE JUNG, PARK, EUNKYUNG, PARK, HYUNJIN, KIM, IN-WOO, KIM, JI-DUCK, CHO, MIN-JAE, YOON, HONGUL, CHO, SEONG-HEE, LEE, IN YOUNG
Format Patent
LanguageChinese
English
Published 01.12.2009
Subjects
CHEMISTRY
HETEROCYCLIC COMPOUNDS
HUMAN NECESSITIES
HYGIENE
MEDICAL OR VETERINARY SCIENCE
METALLURGY
ORGANIC CHEMISTRY
PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS
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Summary:The present invention relates to a novel benzoxazine benzimidazole derivative of formula (1) as an antagonist against a vanilloid receptor-1, a pharmaceutical composition comprising the same as an active ingredient, and a use thereof. The benzoxazine benzimidazole derivative of the present invention may be useful for preventing or treating a disease associated with antagonistic activity of vanilloid receptor-1: wherein, R1, R2, R3, R3', Q1, Q2, Q3 and Q4 have same meanings as defined in the specification.
Bibliography:Application Number: TW200998112800