DERIVATIVES OF QUINOLINECARBOXYLIC AND BORIC ACID ANHYDRIDE AND PROCESS OF PRODUCING THEM

PCT No. PCT/HU88/00018 Sec. 371 Date Dec. 2, 1988 Sec. 102(e) Date Dec. 2, 1988 PCT Filed Apr. 8, 1988 PCT Pub. No. WO88/07998 PCT Pub. Date Oct. 20, 1988.The invention relates to new quinoline-3-carboxylic acid anhydride intermediates of the Formula I (I) wherein R stands for cyclopropyl, a group o...

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Main Authors VASVARI LELLE, BALOGH MARIA, HORVATH AGNES, MARMAROSI KATALIN, HERMECZ ISTVAN, PAJOR ANIKO, KERESZTURI GEZA, RITLI PETER, SIPOS JUDIT
Format Patent
LanguageEnglish
Published 05.11.1997
Edition6
Subjects
ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAININGELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN,SULFUR, SELENIUM OR TELLURIUM
CHEMISTRY
HETEROCYCLIC COMPOUNDS
HUMAN NECESSITIES
HYGIENE
MEDICAL OR VETERINARY SCIENCE
METALLURGY
ORGANIC CHEMISTRY
PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS
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Summary:PCT No. PCT/HU88/00018 Sec. 371 Date Dec. 2, 1988 Sec. 102(e) Date Dec. 2, 1988 PCT Filed Apr. 8, 1988 PCT Pub. No. WO88/07998 PCT Pub. Date Oct. 20, 1988.The invention relates to new quinoline-3-carboxylic acid anhydride intermediates of the Formula I (I) wherein R stands for cyclopropyl, a group of the Formula -CH2CR5R6R7 wherein R5, R6 and R7 stand for hydrogen or halogen, or phenyl optionally substituted by 1 or 2 halogen, R1 and R2 stand for halogen, or an aliphatic acyloxy group containing 2 to 6 carbon atoms optionally substituted by halogen, or an aromatic acyloxy group containing 7 to 11 carbon atoms, R3 stands for chlorine or fluorine and R4 stands for hydrogen or fluorine. The compounds of the Formula I are new intermediates for the preparation of known quinoline-3-carbocxylic acids showing antibacterial activity.
Bibliography:Application Number: SK19880002419