PROCESS FOR PREPARING MODULATORS OF P300 AND/OR CBP
A process for producing a compound of the following formula (I) which process comprises: (a) treating a compound of the following formula (5) with a compound of the following formula (6) to generate an intermediate compound of the following formula (7); (b) treating a compound of formula (7) as defi...
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Main Authors | , , , , , , , , |
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Format | Patent |
Language | English |
Published |
27.11.2020
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Subjects | |
Online Access | Get full text |
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Summary: | A process for producing a compound of the following formula (I) which process comprises: (a) treating a compound of the following formula (5) with a compound of the following formula (6) to generate an intermediate compound of the following formula (7); (b) treating a compound of formula (7) as defined above with a compound of the following formula (8); and (c) recovering a compound of formula (I) as defined above. The compound of formula (I) is a promising modulator of p300/CBP activity that has potential utility in treating cancers, including prostate cancer, haematological cancers, bladder cancer and lung cancer. |
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Bibliography: | Application Number: SG20201109919W |