AMINOAZOLE DERIVATIVE

AMINOAZOLE DERIVATIVE A compound, represented by the following formula or 5 a medically acceptable salt thereof, having an effect of regulating the activity of an androgen receptor. In the formula, X represents S, O; Z represents (R a)n-A-(CR 13 R14 )0- 1-(CR 11 R12 )0-1-; A represents aryl, heteroa...

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Main Authors HOSODA, Shinnosuke, UNOKI, Gen, WATANABE, Hidekazu, HORIE, Kyohei, SASAKI, Kosuke, YOKOYAMA, Emi, SHIBATA, Jun, TAKAGI, Kenichiro
Format Patent
LanguageEnglish
Published 28.06.2018
Subjects
ACYCLIC OR CARBOCYCLIC COMPOUNDS
CHEMISTRY
HETEROCYCLIC COMPOUNDS
HUMAN NECESSITIES
HYGIENE
MEDICAL OR VETERINARY SCIENCE
METALLURGY
ORGANIC CHEMISTRY
PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS
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Summary:AMINOAZOLE DERIVATIVE A compound, represented by the following formula or 5 a medically acceptable salt thereof, having an effect of regulating the activity of an androgen receptor. In the formula, X represents S, O; Z represents (R a)n-A-(CR 13 R14 )0- 1-(CR 11 R12 )0-1-; A represents aryl, heteroaryl; R 1 represents alkyl, cycloalkyl, alkenyl, alkynyl, 10 alkoxyalkyl, aryl, arylalkyl, heterocycle, heterocyclic alkyl; R 2 represents hydrogen, halogen, alkyl, cycloalkyl, phenyl; R3 represents hydrogen, halogen, alkyl, cycloalkyl, alkoxyalkyl, alkenyl, alkynyl, cycloalkenyl, aryl, arylalkyl, heterocycle, heterocyclic alkyl, acyl, 15 cycloalkylcarbonyl, benzoyl, spiroalkyl, adamantyl, silyl, R 31 R32 NCO-; R 4 and R 5 represent hydrogen, halogen, alkyl, phenyl, and cycloalkyl. [Chem. 1] 20 [No Suitable Figure]
Bibliography:Application Number: SG20181104359S