1-PHENYL-1-CYCLOPENTYL-4-PIPERIDINO-2-BUTYNE-1-OL HYDROCHLORIDE (PENTIFIN) ELICITING M4 CHOLINE-BLOCKING ACTIVITY
FIELD: organic chemistry, pharmacy. SUBSTANCE: invention proposes a new agent with expressed selective blocking activity with regards to muscarinic receptors of subtype M4 taking part in control over the formation of cAMP and in activation of peptides Gi/Go. Agent represents 1-phenyl-1-cyclopentyl-4...
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Main Authors | , , , , , , , |
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Format | Patent |
Language | English Russian |
Published |
27.02.2004
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Edition | 7 |
Subjects | |
Online Access | Get full text |
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Summary: | FIELD: organic chemistry, pharmacy. SUBSTANCE: invention proposes a new agent with expressed selective blocking activity with regards to muscarinic receptors of subtype M4 taking part in control over the formation of cAMP and in activation of peptides Gi/Go. Agent represents 1-phenyl-1-cyclopentyl-4-piperidino-2-butyne-1-ol (pentifin) of the formula (I) known early as an agent used in treatment of Parkinson's disease. EFFECT: valuable medicinal properties of agent, expanded assortment of agents of indicated designation. 1 tbl, 1 ex |
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Bibliography: | Application Number: RU20020127885 |