ARYLALIPHATIC AMINOAMIDES OF PHENOXYACETIC ACID OR SUBSTITUTED PHENOXYACETIC ACIDS HAVING LOCAL-ANESTHETIC AND ANALGETIC ACTIVITY

• Main Authors: GOLOVKOV P.V, LUKASHOVA L.A, BORISOVA E.JA, TEREKHOVA O.A, KLOCHKOVA A.R, BORISOVA N.JU, POPOVA I.L, ELISEEVA I.A, ARZAMASTSEV E.V, CHERKASHIN M.I
• Format: Patent
• Language: English
• Published: 27.03.1999
• Edition: 6
• Subjects: ACYCLIC OR CARBOCYCLIC COMPOUNDS; CHEMISTRY; HUMAN NECESSITIES; HYGIENE; MEDICAL OR VETERINARY SCIENCE; METALLURGY; ORGANIC CHEMISTRY; PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES; SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS

FIELD: medicine. SUBSTANCE: present invention describes biologically active compounds, more particularly arylaliphatic aminoazides of general formula I: wherein when R is CH2OC6H5,, then R1 is NC4H8O, and n is 4,5, 6 and 7; R1 is NC5H10,, and n is 4,5,6 and 7; when R is CH2OC6H4CH3-4, then R1 is N(CH3)2,, and n is 4,5,6 and 7; when R is CH2OC6H4CH3-2,, then R1 is NC5H10, and n is 4,5,6 and 7; when R is CH2OC6H4OCH3-2, then R1 is N(CH3)2, and n is 4,5,6 and 7; when R is CH2OC6H4NO2-4, then R1 is N(C2H5)2, and n is 4,5,6,7; when R is CH2OC6H4F-4, then R1 is NC5H10, and n is 4,5,6,7; when R is CH2OC6H4Br-4, then R1 is N(CH3)2,, and n is 4,5,6,7; when R is CH2OC6H4Cl-2, then R1 is NC5H10, and n is 4,5,6 and 7; R1 is N(CH3)2 and n is 4,5,6 and 7; when R is CH2OC6H4Cl-3, then R1 is NC4H8O, and n is 4,5,6 and 7; when R1 is N(CH3)2 and n is 4,5,6 and 7; when R is CH2OC6H4Cl-4, then R1/ is NC4H8O, and n is 4,5,6 and 7; when R1 is NC5H10, and n is 4,5,6,7; when R is CH2OC6H3Cl2-2,4, then R1 is N(CH3)2, and n is 4,5,6 and 7; when R1 is NC5H10, and n is 4,5,6 and 7; when R1 is N(C2H5)2, and n is 4,5,6,7; when R1 is NC4H8O and n is 4,5,6,7; when R is CH2</SB