FLUORO-SUBSTITUTED MILBEMYCINS AND AVERMECTINS FOR COMBATTING PARASITES AND INSECTS

Novel avermectin and milbemycin compounds, wherein at least one of the 4a, 5 or 4 sec positions are substituted with a fluoro groups, are prepared by replacement of hydroxy or other suitable leaving group of avermectin and milbemycin compounds with fluorine. The fluoroavermectin and fluoromilbemycin...

Full description

Saved in:
Bibliographic Details
Main Authors FISHER, MICHAEL H, ESKOLA, PHILIP, MROZIK, HELMUT
Format Patent
LanguageEnglish
Published 25.10.1991
Edition5
Subjects
AGRICULTURE
ANIMAL HUSBANDRY
BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES, AS HERBICIDES
CHEMISTRY
DERIVATIVES THEREOF
FISHING
FORESTRY
HETEROCYCLIC COMPOUNDS
HUMAN NECESSITIES
HUNTING
HYGIENE
MEDICAL OR VETERINARY SCIENCE
METALLURGY
NUCLEIC ACIDS
NUCLEOSIDES
NUCLEOTIDES
ORGANIC CHEMISTRY
PEST REPELLANTS OR ATTRACTANTS
PLANT GROWTH REGULATORS
PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTSTHEREOF
SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS
SUGARS
TRAPPING
Online AccessGet full text

Cover

More Information
Summary:Novel avermectin and milbemycin compounds, wherein at least one of the 4a, 5 or 4 sec positions are substituted with a fluoro groups, are prepared by replacement of hydroxy or other suitable leaving group of avermectin and milbemycin compounds with fluorine. The fluoroavermectin and fluoromilbemycin compounds have utility as anti-parasitic agents and as highly potent insecticides against agricultural pests.
Bibliography:Application Number: NZ19890228866