ANTAGONISTS OF THE VANILLOID RECEPTOR SUBTYPE 1 (VR1) AND USES THEREOF

ANTAGONISTS OF THE VANILLOED RECEPTOR SUBTYPE I (VRI) AND USES THEIREOF THE PRESENT INVENTION IS DIRECTED TO COMPOUNDS OF FORMULA (1), WHEREIN VARIABLES X', X', Y, 5 R", R IB, R?I, R2B , AL, A2,A3, AND A4ARE AS DEFINED IN THE DESCRIPTION, AND MEDIODS OF USE TO TREAT PAIN, RIEUROPADIIC...

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Main Authors GOMTSYAN, ARTHUR R, KOENIG, JOHN R, BROWN, BRIAN S, LEE, CHIH-HUNG
Format Patent
LanguageEnglish
Published 29.08.2011
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Summary:ANTAGONISTS OF THE VANILLOED RECEPTOR SUBTYPE I (VRI) AND USES THEIREOF THE PRESENT INVENTION IS DIRECTED TO COMPOUNDS OF FORMULA (1), WHEREIN VARIABLES X', X', Y, 5 R", R IB, R?I, R2B , AL, A2,A3, AND A4ARE AS DEFINED IN THE DESCRIPTION, AND MEDIODS OF USE TO TREAT PAIN, RIEUROPADIIC PAIN, ALLODYNIA, PAIN ASSOCIATED WITH FIFFLAINMATION OR AN INFLAIRMIATORY DISEASE, INFLARNMATORY HYPERALGESIA, BLADDER OVERACTIVITY, AND URINARY INCONTINENCE. COR 1 B AL R 1 BR A3
Bibliography:Application Number: MY2008PI04102