NEW DERIVATIVES OF ARTEMISININ , AND THEIR USES IN THE TREATMENT OF MALARIA

A SUBJECT OF THE PRESENT INVENTION IS NEW ARTEMISININ DERIVATIVES, OF FOLLOWING GENERAL FORMULA (I);IN WHICH;@-A AND B REPRESENT A SINGLE OR A DOUBLE BOND,@-N1 AND N2 REPRESENT 0 OR 1,@R1 REPRESENTS A FLUOROALKYL GROUP OR A FLUOROARL GROUP,@-R2 REPRESENTS A HYDROGEN ATOM, OR A HALOGEN ATOM, OR A GRO...

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Main Authors BONNET-DELPON, DANIELE, GRELLEPOIS, FABIENNE, MAGUEUR, GUILLAUME, OUREVITCH, MICHELE, BEGUE, JEAN-PIERRE, CROUSSE, BENOIT, CHORKI, FATIMA
Format Patent
LanguageEnglish
Published 30.09.2009
Subjects
CHEMISTRY
HETEROCYCLIC COMPOUNDS
HUMAN NECESSITIES
HYGIENE
MEDICAL OR VETERINARY SCIENCE
METALLURGY
ORGANIC CHEMISTRY
SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS
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Summary:A SUBJECT OF THE PRESENT INVENTION IS NEW ARTEMISININ DERIVATIVES, OF FOLLOWING GENERAL FORMULA (I);IN WHICH;@-A AND B REPRESENT A SINGLE OR A DOUBLE BOND,@-N1 AND N2 REPRESENT 0 OR 1,@R1 REPRESENTS A FLUOROALKYL GROUP OR A FLUOROARL GROUP,@-R2 REPRESENTS A HYDROGEN ATOM, OR A HALOGEN ATOM, OR A GROUP, IF APPROPRIATE IONISABLE, MAKING IT POSSIBLE TO RENDER SAID COMPOUNDS OF FORMULA (I) WATER-SOLUBLE,@-R3 REPRESENTS A GROUP, IF APPROPRIATES IONISIBLE, MAKING IT POSSIBLE TO RENDER SAID COMPOUNDS OF FORMULA (I) WATER-SOLUBLE,@-R4 REPRESENTS H OR OH.THE INVENTION ALSO RELATES TO THE PROCESS BY WHICH THEY ARE OBTAINED, AND THEIR USES IN PHARMACEUTICAL COMPOSITION INTENDED FOR THE TREATMENT OF MALARIA.
Bibliography:Application Number: MY2002PI03936