3,3-DIARYLPROPYLAMINES, THEIR USE AND PREPARATION

• Main Authors: EMOND, RIKARD, SJOBERG, BIRGER, RINGBERG, ERIK, VAGBERG, JAN, HARALDSSON, MARTIN, BEIERLEIN, KATARINA, JOHNSSON, ROLF
• Format: Patent
• Language: English
• Published: 30.04.2007
• Subjects: ACYCLIC OR CARBOCYCLIC COMPOUNDS; CHEMISTRY; HETEROCYCLIC COMPOUNDS; HUMAN NECESSITIES; HYGIENE; MEDICAL OR VETERINARY SCIENCE; METALLURGY; ORGANIC CHEMISTRY; PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES; SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS

THE INVENTION RELATES TO NOVEL COMPOUNDS OF FORMULA (1): WHEREIN R1, R2, R3, R4, R5, R6, R7 AND AR ARE AS DEFINED IN CLAIM 1, THEIR SALTS WITH PHYSIOLOGICALLY ACCEPTABLE ACIDS AND, WHEN THE COMPOUNDS CAN BE IN THE FORM OF OPTICAL ISOMERS, THE RACEMIC MIXTURE AND THE INDIVIDUAL ENANTIOMERS. THE COMPOUNDS HAVE ANTICHOLINERGIC ACTIVITY, AND THE INVENTION ALSO RELATES TO THE COMPOUNDS OF FORMULA 1 FOR USE AS THERAPEUTICALLY ACTIVE SUBSTANCES, PHARMACEUTICAL COMPOSITIONS CONTAINING COMPOUNDS OF FORMULA 1, THE USE OF THE COMPOUNDS OF FORMULA 1 FOR PREPARING ANTICHOLINERGIC DRUGS, THE USE OF THE COMPOUNDS OF FORMULA 1 FOR TREATING URINARY INCONTINENCE, AND METHODS FOR PREPARING THE COMPOUNDS OF FORMULA 1.