ANTAGONISTS TO THE VANILLOID RECEPTOR SUBTYPE 1 (VR1) AND USES THEREOF

Compounds having formula (I) or formula (II), or a pharmaceutically acceptablesalt, prodrug, or salt of a prodrug thereof, wherein A, N, X, Y, R1, R2and R3 are as defined in the specification. These compounds are particularlyuseful in the treatment of pain, inflammatory hyperalgesia, and urinary dys...

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Bibliographic Details
Main Authors RYAN G. KEDDY, CHIH-HUNG LEE, BRIAN S. BROWN, RICHARD J. PERNER, JOHN R. KOENIG
Format Patent
LanguageEnglish
Spanish
Published 25.07.2007
Subjects
CHEMISTRY
HETEROCYCLIC COMPOUNDS
HUMAN NECESSITIES
HYGIENE
MEDICAL OR VETERINARY SCIENCE
METALLURGY
ORGANIC CHEMISTRY
PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS
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Summary:Compounds having formula (I) or formula (II), or a pharmaceutically acceptablesalt, prodrug, or salt of a prodrug thereof, wherein A, N, X, Y, R1, R2and R3 are as defined in the specification. These compounds are particularlyuseful in the treatment of pain, inflammatory hyperalgesia, and urinary dysfunctions,such as bladder overactivity and urinary incontinence. Compuestos que tienen la formula (I) o la formula (II), o una sal, profarmaco, o sal de un profarmaco del mismo farmaceuticamente aceptables, en donde A, N, X, Y, R1, R2 y R3 son como se definen en la especificacion. Estos compuestos son particularmente utiles en el tratamiento del dolor, hiperalgesia inflamatoria, y disfuncion urinaria, tal como superactividad de la vejiga e incontinencia urinaria.
Bibliography:Application Number: MX20070006846