MACROLIDE COMPOUNDS, THEIR PREPARATION AND THEIR USE

• Main Authors: TANAKA, KEIKO, KAJINO, HISAKI, IWADO, SEIGO, YANAI, TOSHIAKI, OKAZAKI, TAKAO, TAKAHASHI, SHUJI
• Format: Patent
• Language: English; Korean
• Published: 30.09.1996
• Edition: 6
• Subjects: AGRICULTURE; ANIMAL HUSBANDRY; BEER; BIOCHEMISTRY; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES, AS HERBICIDES; CHEMISTRY; COMPOSITIONS THEREOF; CULTURE MEDIA; DERIVATIVES THEREOF; ENZYMOLOGY; FERMENTATION OR ENZYME-USING PROCESSES TO SYNTHESISE A DESIREDCHEMICAL COMPOUND OR COMPOSITION OR TO SEPARATE OPTICAL ISOMERSFROM A RACEMIC MIXTURE; FISHING; FORESTRY; HETEROCYCLIC COMPOUNDS; HUMAN NECESSITIES; HUNTING; HYGIENE; MEDICAL OR VETERINARY SCIENCE; METALLURGY; MICROBIOLOGY; MICROORGANISMS OR ENZYMES; MUTATION OR GENETIC ENGINEERING; NUCLEIC ACIDS; NUCLEOSIDES; NUCLEOTIDES; ORGANIC CHEMISTRY; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS; PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES; PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTSTHEREOF; PROPAGATING, PRESERVING OR MAINTAINING MICROORGANISMS; SPIRITS; SUGARS; TRAPPING; VINEGAR; WINE

없음. Compounds with acaricidal, insecticidal and anthelmintic activities have the formula: wherein: -X-Y- is -CH2-CH2-, -CH2-CHOH-, -CH=CH-, or -CH2-C(=O)-; R is a methyl group, an ethyl group, an isopropyl group, a sec-butyl group or a group of formula -C(CH3)=CHR in which R is a methyl group, an ethyl group or an isopropyl group; R represents a group of formula -(CH2)n-C(R )=C(R )(R ) in which n is 0, 1 or 2, R and R each is a hydrogen atom or a methyl group and R is a hydrogen atom, a C1-4 alkyl group, a phenyl group or a phenyl group substituted with at least one substituent selected from halogen, methyl and/or nitro substituents; R is a hydrogen atom, a methyl group, a hydroxy-protecting group, an ester-forming carboxylic acid residue, or an ester-forming carbonic acid residue; and R is a hydrogen atom or an alpha -L-oleandrosyl- alpha -L-oleandrosyloxy group, with the proviso that R represents a hydrogen atom when the group R is a methyl group, an ethyl group, or a group of formula -C(CH3)=CHR in which R is a methyl group, an ethyl group or an isopropyl group.