PROCESS FOR PREPARING 5,9-B-DISUBSTITUTED 2-TETRAHY-DROFURFURYL-6,7-BENZOMORPHANS

Title compds. (I; R = H, Me, acetyl, R1 = Me, Ph), useful sedative, and their acid addition salt were prepd. by alkylation norbenzomorphane II with III (X = neuclephilically eliminable group such as halogen atom of Cl, Br, and I aralkylsulfonyloxy or alkylsulfonyloxy) in the presence of acid binding...

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Bibliographic Details
Main Authors GERHARD WALTHER, HERBERT MERZ, KLAUS STOCKHAUS, ADOLF LANG BEIN
Format Patent
LanguageEnglish
Published 18.09.1979
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Summary:Title compds. (I; R = H, Me, acetyl, R1 = Me, Ph), useful sedative, and their acid addition salt were prepd. by alkylation norbenzomorphane II with III (X = neuclephilically eliminable group such as halogen atom of Cl, Br, and I aralkylsulfonyloxy or alkylsulfonyloxy) in the presence of acid binding agent such as triethylamine, dicyclohexylethylamine, etc.
Bibliography:Application Number: KR19750001720