세레블론 결합 화합물, 이의 조성물, 및 이에 의한 치료 방법

하기 구조를 갖는 피페리딘 디온 화합물, 피페리딘 디온 화합물의 유효량을 포함하는 조성물, 및 안드로겐 수용체 매개 질병을 치료 또는 예방하기 위한 방법이 본 명세서에 제공된다: [화학식 I] JPEGpct00106.jpg2479 (상기 식에서, RN, R1, R2, R3, R4, RN, L, V, X, a, m, 및 n은 본 명세서에 정의된 바와 같음). Provided herein are piperidine dione compounds having the following structure:wherein RN, R1, R2, R...

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Main Authors ALEXANDER MATTHEW D, HARRIS III ROY L, HORN EVAN J, DALVIE DEEPAK, PLANTEVIN KRENITSKY VERONIQUE, MAYNE CHRISTOPHER, NORRIS STEPHEN, CORREA MATTHEW D, WHITEFIELD BRANDON W, HANSEN JOSHUA, SAPIENZA JOHN J, GRANT VIRGINIA HEATHER SHARRON, HUANG DEHUA, TEHRANI LIDA
Format Patent
LanguageKorean
Published 27.02.2023
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Abstract 하기 구조를 갖는 피페리딘 디온 화합물, 피페리딘 디온 화합물의 유효량을 포함하는 조성물, 및 안드로겐 수용체 매개 질병을 치료 또는 예방하기 위한 방법이 본 명세서에 제공된다: [화학식 I] JPEGpct00106.jpg2479 (상기 식에서, RN, R1, R2, R3, R4, RN, L, V, X, a, m, 및 n은 본 명세서에 정의된 바와 같음). Provided herein are piperidine dione compounds having the following structure:wherein RN, R1, R2, R3, R4, RN, L, V, X, a, m, and n are as defined herein, compositions comprising an effective amount of a piperidine dione compound, and methods for treating or preventing an androgen receptor mediated disease.
AbstractList 하기 구조를 갖는 피페리딘 디온 화합물, 피페리딘 디온 화합물의 유효량을 포함하는 조성물, 및 안드로겐 수용체 매개 질병을 치료 또는 예방하기 위한 방법이 본 명세서에 제공된다: [화학식 I] JPEGpct00106.jpg2479 (상기 식에서, RN, R1, R2, R3, R4, RN, L, V, X, a, m, 및 n은 본 명세서에 정의된 바와 같음). Provided herein are piperidine dione compounds having the following structure:wherein RN, R1, R2, R3, R4, RN, L, V, X, a, m, and n are as defined herein, compositions comprising an effective amount of a piperidine dione compound, and methods for treating or preventing an androgen receptor mediated disease.
Author HUANG DEHUA
HORN EVAN J
SAPIENZA JOHN J
HARRIS III ROY L
WHITEFIELD BRANDON W
PLANTEVIN KRENITSKY VERONIQUE
NORRIS STEPHEN
CORREA MATTHEW D
HANSEN JOSHUA
ALEXANDER MATTHEW D
MAYNE CHRISTOPHER
TEHRANI LIDA
GRANT VIRGINIA HEATHER SHARRON
DALVIE DEEPAK
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– fullname: MAYNE CHRISTOPHER
– fullname: NORRIS STEPHEN
– fullname: CORREA MATTHEW D
– fullname: WHITEFIELD BRANDON W
– fullname: HANSEN JOSHUA
– fullname: SAPIENZA JOHN J
– fullname: GRANT VIRGINIA HEATHER SHARRON
– fullname: HUANG DEHUA
– fullname: TEHRANI LIDA
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Snippet 하기 구조를 갖는 피페리딘 디온 화합물, 피페리딘 디온 화합물의 유효량을 포함하는 조성물, 및 안드로겐 수용체 매개 질병을 치료 또는 예방하기 위한 방법이 본 명세서에 제공된다: [화학식 I] JPEGpct00106.jpg2479 (상기 식에서, RN, R1, R2, R3, R4,...
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SubjectTerms CHEMISTRY
HETEROCYCLIC COMPOUNDS
HUMAN NECESSITIES
HYGIENE
MEDICAL OR VETERINARY SCIENCE
METALLURGY
ORGANIC CHEMISTRY
PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS
Title 세레블론 결합 화합물, 이의 조성물, 및 이에 의한 치료 방법
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