ASK1 SOLID FORMS OF AN ASK1 INHIBITOR
5-(4-시클로프로필-1H-이미다졸-1-일)-N-(6-(4-이소프로필-4H-1,2,4-트리아졸-3-일)피리딘-2-일)-2-플루오로-4-메틸벤즈아미드 (화합물 I)의 결정질 형태를 제조하고, 고체 상태로 특징화하였다. 상기 결정질 형태의 제조 방법 및 사용 방법이 또한 제공된다. Crystalline forms of 5-(4-cyclopropyl-1H-imidazol-1-yl)-N-(6-(4-isopropyl-4H-1,2,4-triazol-3-yl)pyridin-2-yl)-2-fluoro-4-methylbenzamide (Compou...
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Format | Patent |
Language | English Korean |
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23.08.2017
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Abstract | 5-(4-시클로프로필-1H-이미다졸-1-일)-N-(6-(4-이소프로필-4H-1,2,4-트리아졸-3-일)피리딘-2-일)-2-플루오로-4-메틸벤즈아미드 (화합물 I)의 결정질 형태를 제조하고, 고체 상태로 특징화하였다. 상기 결정질 형태의 제조 방법 및 사용 방법이 또한 제공된다.
Crystalline forms of 5-(4-cyclopropyl-1H-imidazol-1-yl)-N-(6-(4-isopropyl-4H-1,2,4-triazol-3-yl)pyridin-2-yl)-2-fluoro-4-methylbenzamide (Compound I) were prepared and characterized in the solid state:Also provided are processes of manufacture and methods of using the crystalline forms. |
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AbstractList | 5-(4-시클로프로필-1H-이미다졸-1-일)-N-(6-(4-이소프로필-4H-1,2,4-트리아졸-3-일)피리딘-2-일)-2-플루오로-4-메틸벤즈아미드 (화합물 I)의 결정질 형태를 제조하고, 고체 상태로 특징화하였다. 상기 결정질 형태의 제조 방법 및 사용 방법이 또한 제공된다.
Crystalline forms of 5-(4-cyclopropyl-1H-imidazol-1-yl)-N-(6-(4-isopropyl-4H-1,2,4-triazol-3-yl)pyridin-2-yl)-2-fluoro-4-methylbenzamide (Compound I) were prepared and characterized in the solid state:Also provided are processes of manufacture and methods of using the crystalline forms. |
Author | CHAN BRENDA J. BURKE LAPINA OLGA VIKTOROVNA ANDRES MARK NOTTE GREGORY CARRA ERNEST A SMOLENSKAYA VALERIYA CHIU ANNA LATHROP STEPHEN P YU LOK HIM |
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Snippet | 5-(4-시클로프로필-1H-이미다졸-1-일)-N-(6-(4-이소프로필-4H-1,2,4-트리아졸-3-일)피리딘-2-일)-2-플루오로-4-메틸벤즈아미드 (화합물 I)의 결정질 형태를 제조하고, 고체 상태로 특징화하였다. 상기 결정질 형태의 제조 방법 및 사용 방법이 또한 제공된다.... |
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Title | ASK1 SOLID FORMS OF AN ASK1 INHIBITOR |
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