13-SUBSTITUTED MIBEMYCIN DERIVATIVES, THE COMPOSITION CONTAINING THEM AND INSECTICIDAL METHOD

• Main Authors: ICHINOSE, REIJI, YANAI, TOSHIAKI, SATO, KAZUO, TAKOSHIBA, HIDEO, TANIZAWA, KINJI, YOKOI, SHINJI
• Format: Patent
• Language: English; Korean
• Published: 15.09.1999
• Edition: 6
• Subjects: AGRICULTURE; ANIMAL HUSBANDRY; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES, AS HERBICIDES; CHEMISTRY; DERIVATIVES THEREOF; FISHING; FORESTRY; HETEROCYCLIC COMPOUNDS; HUMAN NECESSITIES; HUNTING; METALLURGY; NUCLEIC ACIDS; NUCLEOSIDES; NUCLEOTIDES; ORGANIC CHEMISTRY; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS; PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTSTHEREOF; SUGARS; TRAPPING

하기 일반식 (Ⅰ) 인 13 위치에 치환된 밀베마이신 유도체 : (상기 식에서 : R은 메틸, 에틸, 이소프로필 또는 sec-부틸이며; R는 수소 또는 알킬이며; X는 (α-히드록시이미노-또는 α-알콕시이미노-치환된)-아릴메틸 또는 (α-히드록시이미노-또는 α-알콕시이미노-치환된)-헤테로시클릴메틸, N-치환된-아미노페닐 또는 N-치환된-아미노페녹시이며; m은 0 또는 1이며; 그리고 n 도 0 또는 1 이다)는 농업 및 원예학적 구충, 살진드기 및 살충제로서 가치가 있다. 13-Substituted milbemycin derivatives having the formula (I): wherein: R is methyl, ethyl, isopropyl or sec-butyl; R is hydrogen or alkyl; X is ( alpha -hydroxyimino- or alpha -alkoxyimino-substituted)-arylmethyl or ( alpha -hydroxyimino- or alpha -alkoxyimino-substituted)-heterocyclylmethyl, N-substituted-aminophenyl or N-substituted-aminophenoxy; m is 0 or 1; and n is 0 or 1; are valuable as agricultural and horticultural anthelmintic, acaricidal and insecticidal agents.