ISTRADEFYLLINE PREPARATION
To provide a novel formulation with improved dissolution properties of istradefylline.SOLUTION: An oral solid preparation according to one embodiment of the present invention comprises: istradefylline or a pharmaceutically acceptable salt thereof; and hydroxypropylcellulose and/or sucrose fatty acid...
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Format | Patent |
Language | English Japanese |
Published |
28.12.2023
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Abstract | To provide a novel formulation with improved dissolution properties of istradefylline.SOLUTION: An oral solid preparation according to one embodiment of the present invention comprises: istradefylline or a pharmaceutically acceptable salt thereof; and hydroxypropylcellulose and/or sucrose fatty acid ester having a molar substitution degree of 3.SELECTED DRAWING: Figure 3
【課題】イストラデフィリンの溶出性が改善された新規の製剤を提供する。【解決手段】本発明の一態様に係る経口固形製剤は、イストラデフィリンまたはその薬学的に許容される塩と、モル置換度が3のヒドロキシプロピルセルロースおよび/またはショ糖脂肪酸エステルと、を含んでいる。【選択図】図3 |
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AbstractList | To provide a novel formulation with improved dissolution properties of istradefylline.SOLUTION: An oral solid preparation according to one embodiment of the present invention comprises: istradefylline or a pharmaceutically acceptable salt thereof; and hydroxypropylcellulose and/or sucrose fatty acid ester having a molar substitution degree of 3.SELECTED DRAWING: Figure 3
【課題】イストラデフィリンの溶出性が改善された新規の製剤を提供する。【解決手段】本発明の一態様に係る経口固形製剤は、イストラデフィリンまたはその薬学的に許容される塩と、モル置換度が3のヒドロキシプロピルセルロースおよび/またはショ糖脂肪酸エステルと、を含んでいる。【選択図】図3 |
Author | SASAKI TAKASHI OKAMOTO YASUNOBU KATAYAMA TAKESHI HAYASHIDA KAZUKI |
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Snippet | To provide a novel formulation with improved dissolution properties of istradefylline.SOLUTION: An oral solid preparation according to one embodiment of the... |
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Title | ISTRADEFYLLINE PREPARATION |
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