ISTRADEFYLLINE PREPARATION

To provide a novel formulation with improved dissolution properties of istradefylline.SOLUTION: An oral solid preparation according to one embodiment of the present invention comprises: istradefylline or a pharmaceutically acceptable salt thereof; and hydroxypropylcellulose and/or sucrose fatty acid...

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Main Authors OKAMOTO YASUNOBU, HAYASHIDA KAZUKI, SASAKI TAKASHI, KATAYAMA TAKESHI
Format Patent
LanguageEnglish
Japanese
Published 28.12.2023
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Abstract To provide a novel formulation with improved dissolution properties of istradefylline.SOLUTION: An oral solid preparation according to one embodiment of the present invention comprises: istradefylline or a pharmaceutically acceptable salt thereof; and hydroxypropylcellulose and/or sucrose fatty acid ester having a molar substitution degree of 3.SELECTED DRAWING: Figure 3 【課題】イストラデフィリンの溶出性が改善された新規の製剤を提供する。【解決手段】本発明の一態様に係る経口固形製剤は、イストラデフィリンまたはその薬学的に許容される塩と、モル置換度が3のヒドロキシプロピルセルロースおよび/またはショ糖脂肪酸エステルと、を含んでいる。【選択図】図3
AbstractList To provide a novel formulation with improved dissolution properties of istradefylline.SOLUTION: An oral solid preparation according to one embodiment of the present invention comprises: istradefylline or a pharmaceutically acceptable salt thereof; and hydroxypropylcellulose and/or sucrose fatty acid ester having a molar substitution degree of 3.SELECTED DRAWING: Figure 3 【課題】イストラデフィリンの溶出性が改善された新規の製剤を提供する。【解決手段】本発明の一態様に係る経口固形製剤は、イストラデフィリンまたはその薬学的に許容される塩と、モル置換度が3のヒドロキシプロピルセルロースおよび/またはショ糖脂肪酸エステルと、を含んでいる。【選択図】図3
Author SASAKI TAKASHI
OKAMOTO YASUNOBU
KATAYAMA TAKESHI
HAYASHIDA KAZUKI
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Snippet To provide a novel formulation with improved dissolution properties of istradefylline.SOLUTION: An oral solid preparation according to one embodiment of the...
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SubjectTerms HUMAN NECESSITIES
HYGIENE
MEDICAL OR VETERINARY SCIENCE
PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS
Title ISTRADEFYLLINE PREPARATION
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