HYDROXYL, KETO, AND GLUCURONIDE DERIVATIVES OF 3-(4-(7H-PYRROLO[2,3-d]PYRIMIDIN-4-YL)-1H-PYRAZOL-1-YL)-3-CYCLOPENTYLPROPANENITRILE
PROBLEM TO BE SOLVED: To provide new or improved agents which inhibit kinases such as Janus kinases for developing new and more effective pharmaceuticals to treat cancer and other diseases.SOLUTION: The present invention provides hydroxyl, keto, and glucuronide derivatives of 3-(4-(7H-pyrrolo[2,3-d]...
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Main Authors | , , , , , , |
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Format | Patent |
Language | English Japanese |
Published |
21.04.2016
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Subjects | |
Online Access | Get full text |
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Summary: | PROBLEM TO BE SOLVED: To provide new or improved agents which inhibit kinases such as Janus kinases for developing new and more effective pharmaceuticals to treat cancer and other diseases.SOLUTION: The present invention provides hydroxyl, keto, and glucuronide derivatives of 3-(4-(7H-pyrrolo[2,3-d]pyrimidin-4-yl)-1H-pyrazol-1-yl)-3-cyclopentylpropanenitrile.SELECTED DRAWING: None
【課題】癌及び他の疾患を治療する、新しい、より有効な医薬品を開発するために、ヤヌスキナーゼ等のキナーゼを阻害する新しい又は改善された薬剤の提供。【解決手段】本発明は、3−(4−(7H−ピロロ[2,3−d]ピリミジン−4−イル)−1H−ピラゾール−1−イル)−3−シクロペンチルプロパンニトリルのヒドロキシル、ケト及びグルクロニド誘導体を提供する。【選択図】なし |
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Bibliography: | Application Number: JP20150246515 |