ACETYLENE DERIVATIVE AS ANTIINFLAMMATORY MEDICINE/ ANALGESIC
PROBLEM TO BE SOLVED: To provide a compound which acts on the action of a cyclooxygenase enzyme on arachidonic acid to inhibit the biosynthesis of prostaglandins, and is useful for treating or relaxing inflammation-accompanying diseases such as inflammatory arthritis, neurodegeneration and large int...
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| Main Authors | , |
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| Format | Patent |
| Language | English |
| Published |
31.07.2001
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| Edition | 7 |
| Subjects | |
| Online Access | Get full text |
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| Abstract | PROBLEM TO BE SOLVED: To provide a compound which acts on the action of a cyclooxygenase enzyme on arachidonic acid to inhibit the biosynthesis of prostaglandins, and is useful for treating or relaxing inflammation-accompanying diseases such as inflammatory arthritis, neurodegeneration and large intestinal cancer, to provide a medicinal composition thereof, and to provide a method for producing the same. SOLUTION: A compound of represented by the general formula (1), a medicinal composition thereof, and a method for producing the same. For example, a compound having an acetylene group, a pyrazole group and a sulfonamide group and represented by the general formula (2) or (3). |
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| AbstractList | PROBLEM TO BE SOLVED: To provide a compound which acts on the action of a cyclooxygenase enzyme on arachidonic acid to inhibit the biosynthesis of prostaglandins, and is useful for treating or relaxing inflammation-accompanying diseases such as inflammatory arthritis, neurodegeneration and large intestinal cancer, to provide a medicinal composition thereof, and to provide a method for producing the same. SOLUTION: A compound of represented by the general formula (1), a medicinal composition thereof, and a method for producing the same. For example, a compound having an acetylene group, a pyrazole group and a sulfonamide group and represented by the general formula (2) or (3). |
| Author | CHENG HENGMAIO KAWAI AKIYOSHI |
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| Snippet | PROBLEM TO BE SOLVED: To provide a compound which acts on the action of a cyclooxygenase enzyme on arachidonic acid to inhibit the biosynthesis of... |
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| Title | ACETYLENE DERIVATIVE AS ANTIINFLAMMATORY MEDICINE/ ANALGESIC |
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