2-AMINOOXAZOLE DERIVATIVES AS TRPVL ANTAGONISTS USEFUL FOR TREATING PAIN

Compounds of formula (I) wherein R 1 , R 2 , R 4 , and W are defined in the description are TRPV1 antagonists with CNS penetration. Compositions comprising such compounds and methods for treating conditions and disorders using such compounds and compositions are also disclosed.

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Bibliographic Details
Main Authors VASUDEVAN, ANIL, BAYBURT, EROL, K, DAANEN, JEROME, F, KYM, PHILIP R, VOIGHT, ERIC, KOENIG, JOHN R, SCHMIDT, ROBERT, G, GOMTSYAN, ARTHUR, R, PERNER, RICHARD J, KORT, MICHAEL E, DIDOMENICO, STANLEY, JR
Format Patent
LanguageEnglish
Published 12.08.2011
Subjects
CHEMISTRY
HETEROCYCLIC COMPOUNDS
HUMAN NECESSITIES
HYGIENE
MEDICAL OR VETERINARY SCIENCE
METALLURGY
ORGANIC CHEMISTRY
PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS
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Summary:Compounds of formula (I) wherein R 1 , R 2 , R 4 , and W are defined in the description are TRPV1 antagonists with CNS penetration. Compositions comprising such compounds and methods for treating conditions and disorders using such compounds and compositions are also disclosed.
Bibliography:Application Number: HK20110101672