N-(3-Pyrrolidine)-substd. benzamide derivs. - have CNS depressant activity, providing use as psychotropic drugs

Carboxylic acid amide derivs. of formula (I) and salts are new: In (I) R1 and R2 are both lower alkyl or one of R1 and R2 is hydrogen and the other is lower alkyl; X is halogen; R3 is lower alkoxy; R4 is lower alkyl. (I) are useful as psychotropic drugs owing ot their strong CNS depressant activity....

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Bibliographic Details
Main Author MUTSUO TAKASHIMA, SUMIO IWANAMI ET SHINJI USUDA
Format Patent
LanguageEnglish
French
Published 18.07.1980
Subjects
CHEMISTRY
HETEROCYCLIC COMPOUNDS
METALLURGY
ORGANIC CHEMISTRY
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Summary:Carboxylic acid amide derivs. of formula (I) and salts are new: In (I) R1 and R2 are both lower alkyl or one of R1 and R2 is hydrogen and the other is lower alkyl; X is halogen; R3 is lower alkoxy; R4 is lower alkyl. (I) are useful as psychotropic drugs owing ot their strong CNS depressant activity. (I) can be administered orally or parenterally in the form of tablets, capsules, powders, sirups, suppositories or injectable solns. at daily doses of 1-200 mg for adults. La présente invention concerne de nouveaux dérivés de la benzamide. Les dérivés de la benzamide sont représentés par la formule :
Bibliography:Application Number: FR19780036264