SUBSTITUTED INDOLES AND METHODS OF USE THEREOF
The present disclosure provides substituted indole compounds of Formula I: (I) and the pharmaceutically acceptable salts and solvates thereof, wherein R1a, R1e, G1, G2, Q1, Q2, Q3, and (II) are defined as set forth in the specification. The present disclosure is also directed to the use of compounds...
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| Main Authors | , , , , , , , |
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| Format | Patent |
| Language | English French German |
| Published |
23.06.2021
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| Subjects | |
| Online Access | Get full text |
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| Abstract | The present disclosure provides substituted indole compounds of Formula I: (I) and the pharmaceutically acceptable salts and solvates thereof, wherein R1a, R1e, G1, G2, Q1, Q2, Q3, and (II) are defined as set forth in the specification. The present disclosure is also directed to the use of compounds of Formula I to treat a disease, disorder, or condition such as cancer in a subject. |
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| AbstractList | The present disclosure provides substituted indole compounds of Formula I: (I) and the pharmaceutically acceptable salts and solvates thereof, wherein R1a, R1e, G1, G2, Q1, Q2, Q3, and (II) are defined as set forth in the specification. The present disclosure is also directed to the use of compounds of Formula I to treat a disease, disorder, or condition such as cancer in a subject. |
| Author | HARVEY, Darren Martin CAMPBELL, John DUNCAN, Kenneth LAMPE, John THOMENIUS, Michael FOLEY, Megan Alene Cloonan MUNCHHOF, Michael John REITER, Lawrence Alan |
| Author_xml | – fullname: FOLEY, Megan Alene Cloonan – fullname: LAMPE, John – fullname: REITER, Lawrence Alan – fullname: DUNCAN, Kenneth – fullname: MUNCHHOF, Michael John – fullname: HARVEY, Darren Martin – fullname: THOMENIUS, Michael – fullname: CAMPBELL, John |
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| DocumentTitleAlternate | SUBSTITUIERTE INDOLE UND VERFAHREN ZUR VERWENDUNG DAVON INDOLES SUBSTITUÉS ET PROCÉDÉS D'UTILISATION ASSOCIÉS |
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| Notes | Application Number: EP20190849109 |
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| RelatedCompanies | Epizyme, Inc |
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| Snippet | The present disclosure provides substituted indole compounds of Formula I: (I) and the pharmaceutically acceptable salts and solvates thereof, wherein R1a,... |
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| Title | SUBSTITUTED INDOLES AND METHODS OF USE THEREOF |
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