PIPERAZINE DERIVATIVE

[Problem] To provide a compound useful as an MCreceptor agonist. [Solution] The present inventors have made studies on MCreceptor agonists. As a result, it is confirmed that a piperazine derivative has an MCreceptor agonist activity, which leads to the accomplishment of the present invention. The pi...

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Bibliographic Details
Main Authors MORITOMO, Hiroyuki, SUGANE, Takashi, YAMASHITA, Daisuke, HOSOGAI, Naomi, ASAI, Norio
Format Patent
LanguageEnglish
French
German
Published 04.03.2020
Subjects
CHEMISTRY
HETEROCYCLIC COMPOUNDS
HUMAN NECESSITIES
HYGIENE
MEDICAL OR VETERINARY SCIENCE
METALLURGY
ORGANIC CHEMISTRY
PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS
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Summary:[Problem] To provide a compound useful as an MCreceptor agonist. [Solution] The present inventors have made studies on MCreceptor agonists. As a result, it is confirmed that a piperazine derivative has an MCreceptor agonist activity, which leads to the accomplishment of the present invention. The piperazine derivative according to the present invention has an MCreceptor agonist activity, and therefore can be used as a prophylactic or therapeutic agent for disturbance of urination in bladder and urinary tract diseases, particularly underactive bladder, hypotonic bladder, acontractile bladder, detrusor underactivity, neurogenic bladder, urethral relaxation failure, detrusor-sphincter dyssynergia and prostatic hyperplasia.
Bibliography:Application Number: EP20170830975