AMINOAZOLE DERIVATIVE

A compound, represented by the following formula or a medically acceptable salt thereof, having an effect of regulating the activity of an androgen receptor. In the formula, X represents S, O; Z represents (R a ) n -A-(CR 13 R 14 ) 0-1 -(CR 11 R 12 ) 0-1 -; A represents aryl, heteroaryl; R 1 represe...

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Main Authors HOSODA, Shinnosuke, UNOKI, Gen, WATANABE, Hidekazu, HORIE, Kyohei, SASAKI, Kosuke, YOKOYAMA, Emi, SHIBATA, Jun, TAKAGI, Kenichiro
Format Patent
LanguageEnglish
French
German
Published 05.08.2020
Subjects
ACYCLIC OR CARBOCYCLIC COMPOUNDS
CHEMISTRY
HETEROCYCLIC COMPOUNDS
HUMAN NECESSITIES
HYGIENE
MEDICAL OR VETERINARY SCIENCE
METALLURGY
ORGANIC CHEMISTRY
PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS
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Summary:A compound, represented by the following formula or a medically acceptable salt thereof, having an effect of regulating the activity of an androgen receptor. In the formula, X represents S, O; Z represents (R a ) n -A-(CR 13 R 14 ) 0-1 -(CR 11 R 12 ) 0-1 -; A represents aryl, heteroaryl; R 1 represents alkyl, cycloalkyl, alkenyl, alkynyl, alkoxyalkyl, aryl, arylalkyl, heterocycle, heterocyclic alkyl; R 2 represents hydrogen, halogen, alkyl, cycloalkyl, phenyl; R3 represents hydrogen, halogen, alkyl, cycloalkyl, alkoxyalkyl, alkenyl, alkynyl, cycloalkenyl, aryl, arylalkyl, heterocycle, heterocyclic alkyl, acyl, cycloalkylcarbonyl, benzoyl, spiroalkyl, adamantyl, silyl, R 31 R 32 NCO-; R 4 and R 5 represent hydrogen, halogen, alkyl, phenyl, and cycloalkyl.
Bibliography:Application Number: EP20160873130