Beta-lactam antibacterial agents, their pharmaceutical compositions and process for their preparation

The compounds of the formula (I): (I) wherein R1 is a hydrogen atom, a trityl group or an acyl group as found in known antibacterially active penicillins or cephalosporins; R2 is a hydrogen atom, a lower alkyl group or an aryl group; R3 is a hydrogen atom, a lower alkyl group, a substituted lower al...

Full description

Saved in:
Bibliographic Details
Main Author PEARSON, MICHAEL JOHN
Format Patent
LanguageEnglish
French
German
Published 19.09.1979
Subjects
CHEMISTRY
HETEROCYCLIC COMPOUNDS
HUMAN NECESSITIES
HYGIENE
MEDICAL OR VETERINARY SCIENCE
METALLURGY
ORGANIC CHEMISTRY
PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS
Online AccessGet full text

Cover

More Information
Summary:The compounds of the formula (I): (I) wherein R1 is a hydrogen atom, a trityl group or an acyl group as found in known antibacterially active penicillins or cephalosporins; R2 is a hydrogen atom, a lower alkyl group or an aryl group; R3 is a hydrogen atom, a lower alkyl group, a substituted lower alkyl or a thiosubstituted lower alkyl group; and R4 is a group such that CO2R4 is a carboxylic acid group or a salt or readily removable ester thereof; are antibiotics. The compounds may be formulated in pharmaceutical compositions. Processes for the preparation of the compounds (I) are also described.
Bibliography:Application Number: EP19790300230