METHOD FOR SYNTHESIZING D3 DOPAMINE RECEPTOR AGONISTS

An improved method for synthesizing a compound according to formula (I) by reaction of a compound of formula (II) with a sulfinamide according to formula (III). The resultant compound is then reduced and hydrolyzed, and optionally alkylated or arylated to arrive at the compound according to formula...

Full description

Saved in:
Bibliographic Details
Main Authors SIELECKI-DZURDZ THAIS MOTRIA, CHO HYUN, KORTAGERE SANDHYA, MI BAOYU
Format Patent
LanguageChinese
English
Published 08.06.2021
Subjects
ACYCLIC OR CARBOCYCLIC COMPOUNDS
CHEMISTRY
HUMAN NECESSITIES
HYGIENE
MEDICAL OR VETERINARY SCIENCE
METALLURGY
ORGANIC CHEMISTRY
PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
Online AccessGet full text

Cover

More Information
Summary:An improved method for synthesizing a compound according to formula (I) by reaction of a compound of formula (II) with a sulfinamide according to formula (III). The resultant compound is then reduced and hydrolyzed, and optionally alkylated or arylated to arrive at the compound according to formula (I). 用于合成根据式(I)的化合物的改进的方法通过使式(II)的化合物与根据式(III)的亚磺酰胺反应然后将所得化合物还原和水解，并且任选地烷基化或芳基化，以得到根据式(I)的化合物。
Bibliography:Application Number: CN201980070988