PRODUCTION METHOD FOR 1-[5-(2-FLUOROPHENYL)-1-(PYRIDIN-3-YLSULFONYL)-1H-PYRROL-3-YL]-N-METHYLMETHANAMINE MONOFUMARATE

The present invention relates to methods for producing 5-(2-fluorophenyl)-1H-pyrrole-3-carboxyaldehyde by formylation and deprotection and producing 1-[5-(2-fluorophenyl)-1-(pyridin-3-ylsulfonyl)-1H-pyrrol-3-yl]-N-methylmethanamine monofumarate by sulfonylation, etc. 本发明涉及基于甲酰化、脱保护反应的5－(2－氟苯基)－1H－吡咯...

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Bibliographic Details
Main Authors OOI ISAO, IWATA MAKOTO
Format Patent
LanguageChinese
English
Published 11.08.2020
Subjects
APPARATUS THEREFOR
CHEMISTRY
GENERAL METHODS OF ORGANIC CHEMISTRY
HETEROCYCLIC COMPOUNDS
HUMAN NECESSITIES
HYGIENE
MEDICAL OR VETERINARY SCIENCE
METALLURGY
ORGANIC CHEMISTRY
PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS
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Summary:The present invention relates to methods for producing 5-(2-fluorophenyl)-1H-pyrrole-3-carboxyaldehyde by formylation and deprotection and producing 1-[5-(2-fluorophenyl)-1-(pyridin-3-ylsulfonyl)-1H-pyrrol-3-yl]-N-methylmethanamine monofumarate by sulfonylation, etc. 本发明涉及基于甲酰化、脱保护反应的5－(2－氟苯基)－1H－吡咯－3－甲醛的制造方法以及基于磺酰基化等的1－[5－(2－氟苯基)－1－(吡啶－3－基磺酰基)－1H－吡咯－3－基]－N－甲基甲胺单富马酸盐的制造。
Bibliography:Application Number: CN201880082979