PYRIDINE-SULFONAMIDE DERIVATIVES AS SIGMA LIGANDS

The present invention relates to new pyridine-sulfonamide derivatives of formula (I') as sigma ligands having a great affinity for sigma receptors, especially the sigma-1 receptor (?1) and/or sigma-2 receptor (?2), as well as to the process for the preparation thereof, to compositions comprisin...

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Bibliographic Details
Main Authors ALONSO-XALMA, MONICA, ALMANSA-ROSALES, CARMEN, CHRISTMANN, UTE, VIRGILI-BERNADO, MARINA
Format Patent
LanguageEnglish
French
Published 03.11.2022
Subjects
CHEMISTRY
HETEROCYCLIC COMPOUNDS
HUMAN NECESSITIES
HYGIENE
MEDICAL OR VETERINARY SCIENCE
METALLURGY
ORGANIC CHEMISTRY
PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
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Summary:The present invention relates to new pyridine-sulfonamide derivatives of formula (I') as sigma ligands having a great affinity for sigma receptors, especially the sigma-1 receptor (?1) and/or sigma-2 receptor (?2), as well as to the process for the preparation thereof, to compositions comprising them, and to their use as medicaments. La présente invention concerne de nouveaux dérivés de pyridine-sulfonamide de formule (I') utilisés en tant que ligands sigma ayant une grande affinité pour les récepteurs sigma, en particulier le récepteur sigma-1 (?1) et/ou un récepteur sigma-2 (?2), ainsi que son procédé de préparation, des compositions les comprenant, ainsi que leur utilisation en tant que médicaments.
Bibliography:Application Number: CA20223217000